Solid-phase synthesis of tetrasubstituted pyrrolo[2,3-d]pyrimidines.
نویسندگان
چکیده
A facile solid phase synthesis of 2,4,6,7-tetrasubstituted pyrrolo[2,3-d]pyrimidines is described. The synthesis involves a highly efficient five-step route starting from resin-bound dimeric peptoids. To demonstrate the versatility of our method, a representative library of 108 tetrasubstituted pyrrolo[2,3-d]pyrimidines of high quality was synthesized.
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ورودعنوان ژورنال:
- Organic & biomolecular chemistry
دوره 10 21 شماره
صفحات -
تاریخ انتشار 2012